Inhibitor | aEC50without pre-incubation of cells (μM) | bEC50with pre-incubation of cells (μM) | Fold-Change in EC50with pre-incubation (aEC50/bEC50) |
---|---|---|---|
4'-Ed4Tc | 1.03 ± 0.45 | 0.37 ± 0.15 | 2.8 |
LFD4C | 0.34 ± 0.02 | 0.16 ± 0.08 | 2.1 |
DDI | 10.2 ± 1.1 | 5.4 ± 0.8 | 1.9 |
D4Tc | 1.08 ± 0.12 | 1.30 ± 0.21 | 0.8 |
FTC | 0.80 ± 0.04 | 1.03 ± 0.23 | 0.8 |
3TC | 0.40 ± 0.02 | 0.53 ± 0.01 | 0.8 |
NVPc | 0.020 ± 0.004 | 0.063 ± 0.04 | 0.3 |
AZTc | 0.018 ± 0.007 | 0.074 ± 0.040 | 0.2 |