Loop | Mutant | Tropism | IC50 | IC50 | MPI |
---|---|---|---|---|---|
FC increase | |||||
Parental clone | Wild type | R5 | 1.56 nM | - | - |
V2 | V169M | R5 | 1.61 nM | 1.03 | 100% |
V3 | L317W | R5 | 1.90 nM | 1.21 | 100% |
V4 | I408T | R5 | 3.16 nM | 2.02 | 94% |
V2-V3 | V169M | R5 | 1.56 nM | 1.57 | 100% |
L317W | |||||
V2-V4 | V169M | R5 | 1.62 nM | 1.03 | 96% |
I408T | |||||
V3-V4 | L317W | R5 | 1.68 nM | 1.07 | 93% |
I408T | |||||
V2-V3-V4 | V169M | R5 | 1.59 nM | 1.01 | 94% |
L317W | |||||
I408T |